(R)-Ozanimod

This intermediate is coupled with a western fragment and converted to the salt in the final stage. (R)-Ozanimod, typically defined as an intermediate leading to the S-enantiomer of Ozanimod, is employed to synthesize Ozanimod hydrochloride by establishing the crucial chiral amine center, often through chiral ruthenium-catalyzed reduction of an imine intermediate or enzymatic resolution.

API Name Ozanimod hydrochloride
CAS No 1306760-85-9
Molecular Formula C23H25ClN4O3
Molecular Weight 440.9 g/mol
Synonyms 5-[3-[(1R)-1-(2-hydroxyethylamino)-2,3-dihydro-1H-inden-4-yl]-1,2,4-oxadiazol-5-yl]-2-propan-2-yloxybenzonitrile;hydrochloride