Gabapentin enacarbil

Gabapentin enacarbil is a carbamate ester that is the N-[1-(isobutyryloxy)ethoxy]carbonyl derivative of [1-(aminomethyl)cyclohexyl]acetic acid. The prodrug for gabapentin, used for treatment of neuropathic pain and restless legs syndrome. Among its listed roles, it functions as a prodrug, an anticonvulsant and a calcium channel blocker. It is a monocarboxylic acid, a carbamate ester, a carboxylic ester and an acetal. Functionally, it is related to gamma-aminobutyric acid and a gabapentin. It is grouped under the following drug class(es): Gabapentinoids. Its therapeutic use is listed as central nervous system (CNS) agents. The directory classifies it as a commercial API with a synthetic source/manufacturing origin. Other names for this substance include Solzira, Horizant and Regnite. Its PubChem CID is 9883933.

CAS No 478296-72-9
Molecular Formula C16H27NO6
Molecular Weight 329.39 g/mol
Synonyms 2-[1-[[1-(2-methylpropanoyloxy)ethoxycarbonylamino]methyl]cyclohexyl]acetic acid

Frequently Asked Questions