Droloxifene citrate

Droloxifene citrate is a selective estrogen receptor modulator structurally related to tamoxifen. It functions as a tissue-specific estrogen agonist and antagonist, exhibiting antiestrogenic activity in breast tissue while maintaining estrogenic effects on bone and lipid metabolism. It appears as a white to off-white crystalline powder, sparingly soluble in water but soluble in organic solvents including ethanol and methanol. The directory classifies it as a discontinued API with a synthetic source/manufacturing origin. Other names for this substance include 3-Hydroxytamoxifen citrate. Its PubChem CID is 3033766.

CAS No 97752-20-0
Molecular Formula C32H37NO9
Molecular Weight 579.6 g/mol
Synonyms 3-[(E)-1-[4-[2-(dimethylamino)ethoxy]phenyl]-2-phenylbut-1-enyl]phenol;2-hydroxypropane-1,2,3-tricarboxylic acid

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