It is typically subjected to Friedel-Crafts acylation followed by deprotection of the methane sulfonyl groups to produce Raloxifene. 4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate (CAS 84449-65-0) is a key protected intermediate in the synthesis of Raloxifene, serving as a bimesylate derivative that protects the hydroxyl groups on the benzothiophene core.
4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate
| API Name | Raloxifene |
|---|---|
| CAS No | 84449-65-0 |
| Molecular Formula | C16H14O6S3 |
| Molecular Weight | 398.5 g/mol |
| Synonyms | [4-(6-methylsulfonyloxy-1-benzothiophen-2-yl)phenyl] methanesulfonate |
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Frequently Asked Questions
It is typically subjected to Friedel-Crafts acylation followed by deprotection of the methane sulfonyl groups to produce Raloxifene. 4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate (CAS 84449-65-0) is a key protected intermediate in the synthesis of Raloxifene, serving as a bimesylate derivative that protects the hydroxyl groups on the benzothiophene core.
The CAS number of 4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate is 84449-65-0.
The molecular formula of 4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate is C16H14O6S3.
The listed molecular weight of 4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate is 398.5 g/mol.
4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate is listed as being used in connection with the following API: Raloxifene.
The listed synonym or IUPAC name for 4-(6-(Methylsulfonyloxy)benzo(b)thiophen-2-yl)phenyl methanesulfonate is [4-(6-methylsulfonyloxy-1-benzothiophen-2-yl)phenyl] methanesulfonate.