Eletriptan

Eletriptan is an N-alkylpyrrolidine, that is N-methylpyrrolidine in which the pro-R hydrogen at position 2 is replaced by a {5-[2-(phenylsulfonyl)ethyl]-1H-indol-3-yl}methyl group. Among its listed roles, it functions as a serotonergic agonist, a vasoconstrictor agent and a non-steroidal anti-inflammatory drug. It belongs to the class of indoles, a N-alkylpyrrolidine and a sulfone. It is the conjugate base of eletriptan(1+). It is grouped under the following drug class(es): Serotonin agents and Triptans. Its therapeutic use is listed as analgesics and central nervous system (CNS) agents. The directory classifies it as a commercial API with a synthetic source/manufacturing origin. Other names for this substance include Relpax and eletriptanum. Its PubChem CID is 77993.

CAS No 143322-58-1
Molecular Formula C22H26N2O2S
Molecular Weight 382.5 g/mol
Synonyms 5-[2-(benzenesulfonyl)ethyl]-3-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-1H-indole

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