Its specific spatial arrangement (stereochemistry) is essential for diltiazem’s therapeutic activity, making this glycidic ester vital for creating the correct, active form of the final drug. Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate, specifically the (2R,3S) stereoisomer, is a crucial chiral intermediate (or building block) in the industrial synthesis of diltiazem, a widely used calcium channel blocker for treating hypertension and angina.
Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate
| API Name | Diltiazem |
|---|---|
| CAS No | 42245-42-1 |
| Molecular Formula | C11H12O4 |
| Molecular Weight | 208.21 g/mol |
| Synonyms | methyl 3-(4-methoxyphenyl)oxirane-2-carboxylate |
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Frequently Asked Questions
Its specific spatial arrangement (stereochemistry) is essential for diltiazem's therapeutic activity, making this glycidic ester vital for creating the correct, active form of the final drug. Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate, specifically the (2R,3S) stereoisomer, is a crucial chiral intermediate (or building block) in the industrial synthesis of diltiazem, a widely used calcium channel blocker for treating hypertension and angina.
The CAS number of Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate is 42245-42-1.
The molecular formula of Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate is C11H12O4.
The listed molecular weight of Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate is 208.21 g/mol.
Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate is listed as being used in connection with the following API: Diltiazem.
The listed synonym or IUPAC name for Methyl 3-(4-methoxyphenyl)-2-oxiranecarboxylate is methyl 3-(4-methoxyphenyl)oxirane-2-carboxylate.