It functions as a protected indole building block, facilitating the attachment of the piperidinyl moiety. The tert-butyl carboxylate (Boc) group allows for further functionalization, with the 4-formyl group serving as a site for coupling in the synthesis of the final drug substance. Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is a key pharmaceutical intermediate, often employed to synthesize Iptacopan (a Factor B inhibitor for paroxysmal nocturnal hemoglobinuria).
Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate
| API Name | Iptacopan |
|---|---|
| CAS No | 1481631-51-9 |
| Molecular Formula | C16H19NO4 |
| Molecular Weight | 289.33 g/mol |
| Synonyms | tert-butyl 4-formyl-5-methoxy-7-methylindole-1-carboxylate |
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Frequently Asked Questions
It functions as a protected indole building block, facilitating the attachment of the piperidinyl moiety. The tert-butyl carboxylate (Boc) group allows for further functionalization, with the 4-formyl group serving as a site for coupling in the synthesis of the final drug substance. Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is a key pharmaceutical intermediate, often employed to synthesize Iptacopan (a Factor B inhibitor for paroxysmal nocturnal hemoglobinuria).
The CAS number of Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is 1481631-51-9.
The molecular formula of Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is C16H19NO4.
The listed molecular weight of Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is 289.33 g/mol.
Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is listed as being used in connection with the following API: Iptacopan.
The listed synonym or IUPAC name for Tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylate is tert-butyl 4-formyl-5-methoxy-7-methylindole-1-carboxylate.