It is generally condensed with 3-(S)-(+)-(1-carbamoyl-1,1-diphenylmethyl)pyrrolidine (or its derivatives) via nucleophilic substitution, typically in the presence of a base, to form the active API. 5-(2-Chloroethyl)-2,3-dihydrobenzofuran acts as a key intermediate in the synthesis of Darifenacin by providing the 2-(2,3-dihydrobenzofuran-5-yl)ethyl moiety.
5-(2-Chloroethyl)-2,3-dihydrobenzofuran
| API Name | Darifenacin |
|---|---|
| CAS No | 943034-50-2 |
| Molecular Formula | C10H11ClO |
| Molecular Weight | 182.64 g/mol |
| Synonyms | 5-(2-chloroethyl)-2,3-dihydro-1-benzofuran |
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Frequently Asked Questions
It is generally condensed with 3-(S)-(+)-(1-carbamoyl-1,1-diphenylmethyl)pyrrolidine (or its derivatives) via nucleophilic substitution, typically in the presence of a base, to form the active API. 5-(2-Chloroethyl)-2,3-dihydrobenzofuran acts as a key intermediate in the synthesis of Darifenacin by providing the 2-(2,3-dihydrobenzofuran-5-yl)ethyl moiety.
The CAS number of 5-(2-Chloroethyl)-2,3-dihydrobenzofuran is 943034-50-2.
The molecular formula of 5-(2-Chloroethyl)-2,3-dihydrobenzofuran is C10H11ClO.
The listed molecular weight of 5-(2-Chloroethyl)-2,3-dihydrobenzofuran is 182.64 g/mol.
5-(2-Chloroethyl)-2,3-dihydrobenzofuran is listed as being used in connection with the following API: Darifenacin.
The listed synonym or IUPAC name for 5-(2-Chloroethyl)-2,3-dihydrobenzofuran is 5-(2-chloroethyl)-2,3-dihydro-1-benzofuran.